| Year | Rnd | Ovl | Phase | Player | Drafting Team | Pos | HiLvl | Played | Src | Drafted From | SF | State | AB | 2B | 3B | HR | RBI | SB | BAVG | W | L | ERA | SV | IP | SO | GS |
| 2001 | 3 | 77 | June-Reg | Jose Morales | Minnesota Twins | SS | MLB | 2001-2012 | H | -- | SF | 218 | 12 | 0 | 0 | 21 | 0 | .289 | -- | -- | -- | -- | -- | -- | -- | |
| 2001 | 3 | 78 | June-Reg | Ryan Theriot | Chicago Cubs | IF | MLB | 1999-2012 | C | Louisiana State University | SF | LA | 3246 | 138 | 18 | 17 | 257 | 121 | .281 | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 79 | June-Reg | Chris Flinn | Tampa Bay Rays | P | AAA | 2001-2012 | C | Stony Brook University | SF | NY | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 80 | June-Reg | Lazaro Abreu | Seattle Mariners | C | RK | 2001-2001 | H | Dale (Dale,OK) | SF | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | |
| 2001 | 3 | 81 | June-Reg | Steven Shell | Anaheim Angels | P | MLB | 2001-2011 | H | El Reno (El Reno,OK) | SF | OK | 4 | 0 | 0 | 0 | 0 | 0 | .000 | 2 | 2 | 2.45 | 2 | 55 | 46 | 0 |
| 2001 | 3 | 82 | June-Reg | Mike Hinckley | Montreal Expos | P | MLB | 2001-2011 | H | Moore (Moore,OK) | SF | OK | 1 | 0 | 0 | 0 | 0 | 0 | .000 | 0 | 0 | 1.93 | 0 | 23 | 12 | 0 |
| 2001 | 3 | 83 | June-Reg | Dave Crouthers | Baltimore Orioles | P | AA | 2001-2004 | C | Southern Illinois University-Edwardsville | SF | IL | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 84 | June-Reg | Jeremy Guthrie ** | Pittsburgh Pirates | P | MLB | 2001-2013 | C | Stanford University | SF | CA | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 85 | June-Reg | Matt Ferrara | Kansas City Royals | 3B | A- | 2002-2006 | H | Westminster Academy (Fort Lauderdale,FL) | SF | FL | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 86 | June-Reg | Kirk Saarloos | Houston Astros | P | MLB | 1998-2009 | C | Cal State Fullerton | SF | CA | 41 | 2 | 0 | 0 | 5 | 0 | .073 | 29 | 30 | 5.02 | 2 | 509 | 251 | 73 |
| 2001 | 3 | 87 | June-Reg | Jack Hannahan | Detroit Tigers | 3B | MLB | 2001-2013 | C | University of Minnesota | SF | MN | 1463 | 85 | 4 | 28 | 159 | 6 | .234 | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 88 | June-Reg | Jon Steitz | Milwaukee Brewers | P | A | 2001-2003 | C | Yale University | SF | CT | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 89 | June-Reg | Jake Woods | Anaheim Angels | P | MLB | 2001-2010 | H | Kingsburg (Kingsburg,CA) | SF | -- | -- | -- | -- | -- | -- | -- | 8 | 5 | 4.60 | 1 | 162 | 99 | 8 | |
| 2001 | 3 | 90 | June-Reg | Tagg Bozied | San Diego Padres | IF | AAA | 2000-2011 | C | University of San Francisco | SF | CA | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 91 | June-Reg | Tyrell Godwin | Toronto Blue Jays | OF | MLB | 1998-2007 | C | University of North Carolina | SF | NC | 3 | 0 | 0 | 0 | 0 | 0 | .000 | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 92 | June-Reg | Allen Baxter | Florida Marlins | P | A+ | 2001-2006 | H | Varina (Richmond,VA) | SF | VA | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 93 | June-Reg | Jon Devries | Boston Red Sox | C | AA | 2001-2006 | H | Irvine (Irvine,CA) | SF | CA | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 94 | June-Reg | Jason Frome | Colorado Rockies | OF | A+ | 2001-2004 | C | Indiana State University | SF | IN | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 95 | June-Reg | Chase Wright | New York Yankees | P | MLB | 2001-2012 | H | Iowa Park (Iowa Park,TX) | SF | TX | -- | -- | -- | -- | -- | -- | -- | 2 | 0 | 7.20 | 0 | 10 | 8 | 2 |
| 2001 | 3 | 96 | June-Reg | Alan Moye | Cincinnati Reds | OF | AAA | 2001-2007 | H | Pinetree (Longview,TX) | SF | TX | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 97 | June-Reg | Nick Moran | Cleveland Indians | P | A+ | 2000-2007 | C | Fresno State University | SF | CA | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 98 | June-Reg | Scott Hairston | Arizona Diamondbacks | IF | MLB | 2000-2013 | C | Central Arizona College | SF | AZ | 2197 | 124 | 17 | 95 | 279 | 34 | .247 | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 99 | June-Reg | Tim Merritt | Seattle Mariners | IF | AA | 2001-2004 | C | University of South Alabama | SF | AL | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 100 | June-Reg | David Taylor | Los Angeles Dodgers | P | RK | 2001-2001 | H | South Lake (Groveland,FL) | SF | FL | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 101 | June-Reg | J.T. Stotts | Oakland Athletics | IF | AAA | 2001-2006 | C | Cal State Northridge | SF | CA | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 102 | June-Reg | Lenny DiNardo | New York Mets | P | MLB | 2001-2011 | C | Stetson University | SF | FL | 5 | 0 | 0 | 0 | 0 | 0 | .200 | 10 | 18 | 5.36 | 0 | 257 | 132 | 34 |
| 2001 | 3 | 103 | June-Reg | Jon Zeringue ** | Chicago White Sox | C | AA | 2002-2008 | H | E.D. White (Thibodaux,LA) | SF | LA | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |
| 2001 | 3 | 104 | June-Reg | Joe Mather | St. Louis Cardinals | 3B | MLB | 2001-2013 | H | Mountain Pointe (Phoenix,AZ) | SF | AZ | 493 | 26 | 0 | 14 | 49 | 7 | .219 | 0 | 1 | 7.71 | 0 | 2 | 0 | 0 |
| 2001 | 3 | 105 | June-Reg | Adam Stern | Atlanta Braves | OF | MLB | 1999-2010 | H | St. Thomas Aquinas (London,ON) | SF | 43 | 1 | 0 | 1 | 7 | 2 | .116 | -- | -- | -- | -- | -- | -- | -- | |
| 2001 | 3 | 106 | June-Reg | Julian Benavidez | San Francisco Giants | IF | AA | 2001-2010 | C | Diablo Valley College | SF | CA | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- | -- |